💊 Side Effects of Exemestane – AROMED 25 Human Labs
Exemestane is a steroidal aromatase inhibitor. Unlike non-steroidal types, it binds irreversibly to the enzyme aromatase and permanently reduces estrogen levels. Therefore, it helps block tumor growth, but at the same time increases the chance of side effects.
⚡ How Exemestane Works
Exemestane (ATC L02BG06) lowers circulating estrogen by deactivating the enzyme. As a result, tumor cells receive fewer growth signals. This explains its effectiveness in breast cancer therapy. However, because it alters hormone balance, users must be cautious.
📊 Medical Uses
Doctors prescribe exemestane to postmenopausal women as an additional treatment for breast cancer. Since 1999 it has been available in tablet form (Aromasin®, generics). Although it provides significant benefits, patients often report symptoms similar to menopause (PharmaWiki).
⚠️ Common Side Effects
- 🔥 Hot flashes and sweating
- 🤕 Fatigue, headaches, and insomnia
- 🦴 Joint pain and muscle pain
- 🤢 Nausea and digestive discomfort
- 📉 Loss of bone density with long-term use
Most adverse reactions result directly from reduced estrogen. Moreover, many users describe them as menopause-like symptoms (PharmaWiki).
🏋️ Exemestane in Bodybuilding
In addition to medical use, some athletes misuse exemestane as an anti-estrogen. They want to prevent water retention and gynecomastia during steroid cycles. On the other hand, misuse may intensify health risks and cause hormonal imbalance.
💡 Dosage and Administration
Patients usually take exemestane once daily after a meal. Thanks to its long half-life, one dose ensures stable suppression. Nevertheless, self-medication often increases risks and should be avoided.
❓ FAQ – Side Effects of Exemestane
1. What are the most common side effects?
👉 Hot flashes, joint pain, fatigue, and headaches are frequently reported (PubMed).
2. Can men use exemestane safely?
👉 Some men take it in bodybuilding, but long-term use may lead to bone density loss and hormone imbalance.
3. Does exemestane interact with other drugs?
👉 Yes. Since it is metabolized by CYP3A4, drug interactions are possible. In addition, estrogen therapy cancels its effects.
4. Is exemestane allowed in sports?
👉 No. It is banned as a doping substance in competitive athletics.
Reviews
There are no reviews yet.